SCHEMBL16655920

SCHEMBL16655920

COc1cc(F)cc(-c2nn(C3Cc4ccccc4C3)c3ncncc23)c1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 14/20 0.70
BTK Q06187 13/20 0.70
USP2 O75604 4/20 0.41
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
TSHR P16473 4/20 0.41
CYP2C19 P33261 4/20 0.41
ALDH1A1 P00352 2/20 0.39
CYP2C9 P11712 2/20 0.39
MAPK1 P28482 2/20 0.39
LMNA P02545 1/20 0.39
KDM1A O60341 1/20 0.39
ATR Q13535 2/20 0.38
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16655530 0.82 PIK3CD (1.00) PIK3CDBTKATR
SCHEMBL16656011 0.78 PIK3CD (0.59) PIK3CDBTKATR
SCHEMBL16655325 0.77 PIK3CD (1.00) PIK3CDBTKATR
SCHEMBL16655337 0.71 PIK3CD (0.75) PIK3CDBTKATR
SCHEMBL16655617 0.71 ATR (0.47) PIK3CDBTKATR
SCHEMBL23908620 0.69 PIK3CD (0.77) PIK3CDBTKATR
SCHEMBL16655515 0.69 PIK3CD (0.68) PIK3CDBTK
SCHEMBL16655272 0.68 PIK3CD (1.00) PIK3CDBTKATR
SCHEMBL3610794 0.67 PIK3CD (0.75) PIK3CDBTK
SCHEMBL16655153 0.67 PIK3CD (0.76) PIK3CDBTKATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP claimed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO claimed