SCHEMBL16655617

SCHEMBL16655617

c1ccc2c(c1)CC(n1nc(-c3ccc4[nH]cnc4c3)c3cncnc31)C2

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ATR Q13535 9/20 0.47
PIK3CD O00329 12/20 0.42
BTK Q06187 11/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16655267 0.78 ATR (0.76) ATRPIK3CDBTK
SCHEMBL16656011 0.75 PIK3CD (0.59) ATRPIK3CDBTK
SCHEMBL16655920 0.71 PIK3CD (0.70) ATRPIK3CDBTK
SCHEMBL5083828 0.66 IGF1R (0.51) PIK3CD
SCHEMBL21387779 0.66 QPCT (0.38) BTK
SCHEMBL16655575 0.66 PIK3CD (0.66) ATRPIK3CDBTK
SCHEMBL16655264 0.66 PIK3CD (0.69) ATRPIK3CDBTK
SCHEMBL16655349 0.66 ATR (0.89) ATRPIK3CDBTK
SCHEMBL23123086 0.65 QPCT (0.51)
SCHEMBL16655710 0.65 ATR (0.78) ATRPIK3CDBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP claimed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO claimed