SCHEMBL16656113

SCHEMBL16656113

NC(=O)c1ccc(-c2nn(C3CCCc4ccccc43)c3ncnc([AsH2])c23)cc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 18/20 0.49
PIK3CD O00329 4/20 0.49
ATR Q13535 1/20 0.49
EGFR P00533 1/20 0.46
LCK P06239 1/20 0.41
SRC P12931 1/20 0.41
TEK Q02763 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23908597 0.90 BTK (0.61) BTKPIK3CDATREGFRLCK
SCHEMBL16655959 0.84 BTK (0.68) BTKPIK3CDATREGFRLCK
SCHEMBL16655625 0.80 PIK3CD (0.61) BTKPIK3CDATREGFR
SCHEMBL16665786 0.80 PIK3CD (0.61) BTKPIK3CDATREGFR
SCHEMBL16655939 0.78 PIK3CD (0.69) BTKPIK3CDATREGFRLCK
SCHEMBL16655759 0.76 BTK (0.62) BTKPIK3CDATREGFRLCK
SCHEMBL16655479 0.74 PIK3CD (0.68) BTKPIK3CDATREGFRLCK
SCHEMBL16656048 0.74 PIK3CD (0.75) BTKPIK3CDATREGFRSRC
SCHEMBL16665687 0.74 PIK3CD (0.75) BTKPIK3CDATREGFRSRC
SCHEMBL16655658 0.73 ATR (0.71) BTKPIK3CDATRLCKSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP claimed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO claimed