SCHEMBL16657337

SCHEMBL16657337

Brc1c2ccccc2c(-c2ccc(/C=C/c3ccc(-c4cccc5ccccc45)cc3)cc2)c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
ENPP3 O14638 1/20 0.38
ENPP1 P22413 1/20 0.38
PPARG P37231 5/20 0.36
PPARA Q07869 5/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
PPARD Q03181 1/20 0.36
BACE1 P56817 1/20 0.36
MCL1 Q07820 1/20 0.35
ACMSD Q8TDX5 1/20 0.35
CYP1A2 P05177 1/20 0.35
CHAT P28329 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2252435 0.91 HDAC8 (0.50) HDAC8HDAC6CA12CA1CA2
SCHEMBL29658012 0.91 HDAC8 (0.50) HDAC8HDAC6CA12CA1CA2
SCHEMBL29658013 0.91 HDAC8 (0.50) HDAC8HDAC6CA12CA1CA2
SCHEMBL16657335 0.84 HDAC8 (0.51) HDAC8HDAC6CA12CA1CA2
SCHEMBL4820451 0.82 MAOB (0.42) CA1CHAT
SCHEMBL4820453 0.82 MAOB (0.42) CA1CHAT
SCHEMBL24446252 0.82 CA12 (0.55) HDAC8HDAC6CA12CA1CA2
SCHEMBL28491556 0.80 HDAC8 (0.50) HDAC8HDAC6CA12CA1CA2
SCHEMBL16657315 0.80 MEN1 (0.43) HDAC8HDAC6CA12CA1CA2
SCHEMBL16657317 0.79 KDM4E (0.40) HDAC8HDAC6CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9905774-B2 Organic electronic material GUANGDONG AGLAIA OPTOELECTRONIC MATERIALS CO., LTD (CN) 2018-02-27 US disclosed
US-9871202-B2 Organic electroluminescent device GUANGDONG AGLAIA OPTOELECTRONIC MATERIALS CO., LTD (CN) 2018-01-16 US disclosed
US-20150144898-A1 ORGANIC ELECTROLUMINESCENT DEVICE GUANGDONG AGLAIA OPTOELECTRONIC MATERIALS CO., LTD (CN) 2015-05-28 US disclosed
US-20150144898-A1 ORGANIC ELECTROLUMINESCENT DEVICE GUANGDONG AGLAIA OPTOELECTRONIC MATERIALS CO., LTD (CN) 2015-05-28 US disclosed
US-20150108448-A1 ORGANIC ELECTRONIC MATERIAL GUANGDONG AGLAIA OPTOELECTRONIC MATERIALS CO., LTD (CN) 2015-04-23 US disclosed
US-20150108448-A1 ORGANIC ELECTRONIC MATERIAL GUANGDONG AGLAIA OPTOELECTRONIC MATERIALS CO., LTD (CN) 2015-04-23 US disclosed