SCHEMBL16659435

SCHEMBL16659435

C=CC(=O)Nc1cc(N2CCN(CCO)CC2)ccc1Nc1cc(N(C)C(=O)Nc2c(Cl)c(O)cc(OC)c2Cl)ncn1

nearest known ligand 0.92

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 18/20 0.92
FGFR4 P22455 9/20 0.81
FGFR2 P21802 6/20 0.81
FGFR3 P22607 6/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16655971 0.96 FGFR1 (1.00) FGFR1FGFR4FGFR2FGFR3
SCHEMBL16665254 0.94 FGFR1 (0.92) FGFR1FGFR4FGFR2FGFR3
SCHEMBL20081683 0.91 FGFR1 (0.90) FGFR1FGFR4FGFR2FGFR3
SCHEMBL17740763 0.90 FGFR1 (0.92) FGFR1FGFR4FGFR2FGFR3
SCHEMBL16655902 0.90 FGFR1 (1.00) FGFR1FGFR4FGFR2FGFR3
H3B-6527 SCHEMBL16659467 0.89 FGFR1 (1.00) FGFR1FGFR4FGFR2FGFR3
H3B-6527 SCHEMBL29412748 0.89 FGFR1 (1.00) FGFR1FGFR4FGFR2FGFR3
H3B-6527 SCHEMBL30274661 0.89 FGFR1 (1.00) FGFR1FGFR4FGFR2FGFR3
H3B-6527 SCHEMBL30070526 0.89 FGFR1 (0.99) FGFR1FGFR4FGFR2FGFR3
H3B-6527 SCHEMBL30070306 0.89 FGFR1 (0.99) FGFR1FGFR4FGFR2FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015057938-A1 PYRIMIDINE FGFR4 INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2015-04-23 WO disclosed