SCHEMBL1666023

SCHEMBL1666023

CC1(C)OCCN1C(=O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
HTR2C P28335 1/20 0.49
ALDH1A1 P00352 1/20 0.49
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
CYP2C19 P33261 1/20 0.45
P2RX1 P51575 1/20 0.45
P2RX3 P56373 1/20 0.45
P2RX4 Q99571 1/20 0.45
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10797345 0.79 ALDH1A1 (0.53) MEN1KMT2ANPSR1HTR2CALDH1A1
SCHEMBL12656081 0.78 MEN1 (0.49) MEN1KMT2ANPSR1HTR2CNPC1
SCHEMBL3792418 0.77 MEN1 (0.50) MEN1KMT2ANPSR1HTR2CALDH1A1
SCHEMBL14617627 0.76 HTR2C (0.48) MEN1KMT2ANPSR1HTR2CALDH1A1
SCHEMBL2072822 0.76 MEN1 (0.53) MEN1KMT2ANPSR1HTR2CNPC1
SCHEMBL7245273 0.76 MEN1 (0.49) MEN1KMT2ANPSR1HTR2CALDH1A1
SCHEMBL630773 0.76 MEN1 (0.49) MEN1KMT2ANPSR1HTR2CALDH1A1
SCHEMBL15541400 0.76 ALDH1A1 (0.46) MEN1KMT2ANPSR1HTR2CALDH1A1
SCHEMBL1834783 0.75 HTR2C (0.49) MEN1KMT2ANPSR1HTR2CALDH1A1
SCHEMBL542153 0.75 HTR2C (0.49) MEN1KMT2ANPSR1HTR2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486042-A1 BICYCLIC HETEROCYCLES AND THEIR USE AS CCR2 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-08-15 EP disclosed
WO-2011042399-A1 BICYCLIC HETEROCYCLES AND THEIR USE AS CCR2 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-04-14 WO disclosed