SCHEMBL16660264

SCHEMBL16660264

CC(=N)/C=C(\N)Nc1nc(/C=C/c2ccccc2)nc(Nc2cc(C)n[nH]2)c1[N+](=O)[O-]

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.34
MAPT P10636 5/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
LCK P06239 3/20 0.33
SRC P12931 3/20 0.33
BTK Q06187 2/20 0.33
PTK6 Q13882 2/20 0.33
LYN P07948 1/20 0.33
CSK P41240 1/20 0.33
KMT2A Q03164 4/20 0.33
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.33
MAPK1 P28482 1/20 0.33
GAA P10253 2/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL596609 0.86 MAPT (0.43) ADORA3MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL596608 0.86 MAPT (0.43) ADORA3MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL598052 0.77 IGF1R (0.48) ADORA3MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL598053 0.77 IGF1R (0.48) ADORA3MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL596643 0.76 HTT (0.43) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL596644 0.76 HTT (0.43) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL596637 0.75 LMNA (0.44) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL597006 0.75 AURKA (0.38) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL597007 0.75 AURKA (0.38) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL596636 0.75 LMNA (0.44) MAPTCYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928456-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MIIKANA THERAPEUTICS INC (US) 2015-04-22 EP disclosed