SCHEMBL16660839

SCHEMBL16660839

c1ccc(-c2ccc(-c3nc(-c4ccccc4)c[nH]3)cn2)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.54
DHODH Q02127 1/20 0.44
LDHA P00338 1/20 0.43
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
CYP11B1 P15538 4/20 0.41
CYP11B2 P19099 4/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNA3 P32297 2/20 0.41
MAPK1 P28482 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
DYRK1A Q13627 1/20 0.39
DGAT1 O75907 2/20 0.39
BAZ2B Q9UIF8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2837726 0.95 HPGDS (0.57) HPGDSDHODHLDHAHSD17B1HSD17B2
SCHEMBL2837699 0.89 CYP11B1 (0.51) HPGDSLDHACYP11B1CYP11B2MAPK1
SCHEMBL2838619 0.88 HPGDS (0.50) HPGDSDHODHLDHACYP11B1CYP11B2
SCHEMBL2839049 0.88 GSK3B (0.51) HPGDSLDHACYP11B1CYP11B2
SCHEMBL16661139 0.86 HPGDS (0.41) HPGDSDHODHMAPK1DYRK1ADGAT1
SCHEMBL2314781 0.85 HPGDS (0.50) HPGDSDHODHHSD17B1HSD17B2CYP11B1
SCHEMBL7139559 0.85 HPGDS (0.43) HPGDS
SCHEMBL4847155 0.85 HPGDS (0.43) HPGDS
SCHEMBL528246 0.85 MEN1 (0.46) HPGDSMAPK1
SCHEMBL2834537 0.84 HPGDS (0.52) HPGDSDHODHLDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2862856-A1 AROMATIC HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2015-04-22 EP disclosed