SCHEMBL16664430

SCHEMBL16664430

O=C(C[N+]12CCC(CC1)[C@@H](OC(=O)[C@H](Nc1ccccc1)c1ccc(F)cc1)C2)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 16/20 0.41
CHRM2 P08172 5/20 0.41
CHRM1 P11229 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP2D6 P10635 1/20 0.38
PDE2A O00408 1/20 0.38
PDE6D O43924 1/20 0.38
PDE8A O60658 1/20 0.38
PDE5A O76074 1/20 0.38
PDE9A O76083 1/20 0.38
PDE8B O95263 1/20 0.38
PDE6A P16499 1/20 0.38
PDE6G P18545 1/20 0.38
PDE4A P27815 1/20 0.38
PDE6B P35913 1/20 0.38
PDE6C P51160 1/20 0.38
PDE1A P54750 1/20 0.38
PDE1B Q01064 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13240977 1.00 CHRM3 (0.41) CHRM3CHRM2CHRM1NPSR1CYP2D6
Bromide SCHEMBL2485675 0.99 CHRM3 (0.43) CHRM3CHRM2CHRM1NPSR1CYP2D6
SCHEMBL3778319 0.98 CHRM3 (0.41) CHRM3CHRM2CHRM1NPSR1CYP2D6
SCHEMBL13240947 0.96 CHRM3 (0.41) CHRM3CHRM2CHRM1NPSR1CYP2D6
SCHEMBL13240869 0.96 CHRM3 (0.41) CHRM3CHRM2CHRM1NPSR1PDE2A
SCHEMBL3780781 0.96 CHRM3 (0.41) CHRM3CHRM2CHRM1NPSR1PDE2A
SCHEMBL13240907 0.96 CHRM3 (0.41) CHRM3CHRM2CHRM1NPSR1PDE2A
SCHEMBL16649302 0.95 CHRM3 (0.46) CHRM3CHRM2CHRM1NPSR1CYP2D6
SCHEMBL13240958 0.95 CHRM3 (0.46) CHRM3CHRM2CHRM1NPSR1CYP2D6
SCHEMBL16664377 0.95 CHRM3 (0.46) CHRM3CHRM2CHRM1NPSR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376489-B1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF CHIESI FARMA SPA (IT) 2015-04-22 EP disclosed