SCHEMBL16665789

SCHEMBL16665789

C=CC(=O)Nc1cc(-c2n[nH]c3ncnc(N)c23)ccc1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 7/20 0.43
SRC P12931 3/20 0.42
JAK1 P23458 2/20 0.39
MAP2K7 O14733 3/20 0.39
AURKA O14965 1/20 0.39
BTK Q06187 5/20 0.38
ITK Q08881 2/20 0.38
ERBB3 P21860 1/20 0.38
EGFR P00533 4/20 0.38
PIK3CD O00329 2/20 0.38
ABL1 P00519 2/20 0.38
HCK P08631 2/20 0.38
KDR P35968 2/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CB P42338 2/20 0.38
MTOR P42345 2/20 0.38
PIK3CG P48736 2/20 0.38
EPHB4 P54760 2/20 0.38
PRKDC P78527 2/20 0.38
PI4KB Q9UBF8 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16665788 0.91 SRC (0.42) JAK3SRCJAK1MAP2K7AURKA
SCHEMBL23917549 0.79 SRC (0.59) JAK3SRCAURKABTKITK
SCHEMBL16665792 0.79 SRC (0.45) JAK3SRCJAK1MAP2K7AURKA
SCHEMBL21467053 0.78 PIK3CG (0.52) SRCEGFRPIK3CDABL1HCK
SCHEMBL16665742 0.76 PIK3CG (0.41) SRCEGFRPIK3CDABL1HCK
SCHEMBL9010 0.75 PIK3CG (0.54) SRCBTKEGFRPIK3CDABL1
SCHEMBL23917271 0.75 BTK (0.40) JAK3SRCBTKITKEGFR
SCHEMBL21467104 0.73 PIK3CD (0.54) SRCBTKEGFRPIK3CDABL1
SCHEMBL11928101 0.73 PIK3CD (0.56) SRCBTKEGFRPIK3CDABL1
SCHEMBL16665803 0.73 PIK3CD (0.57) SRCBTKEGFRPIK3CDABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO disclosed