SCHEMBL16673186

SCHEMBL16673186

C=Cc1cccc2c1CN(C(=O)OC1CNC(C(=O)OC)C1)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM10 O14672 2/20 0.39
ERBB2 P04626 2/20 0.39
MMP1 P03956 1/20 0.39
PIM1 P11309 1/20 0.34
ABHD6 Q9BV23 2/20 0.34
DPP8 Q6V1X1 7/20 0.33
DPP7 Q9UHL4 7/20 0.33
DPP9 Q86TI2 6/20 0.33
HDAC2 Q92769 2/20 0.32
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
DPP4 P27487 2/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
GAA P10253 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2424560 1.00 ADAM10 (0.39) ADAM10ERBB2MMP1PIM1ABHD6
SCHEMBL13658627 1.00 ADAM10 (0.39) ADAM10ERBB2MMP1PIM1ABHD6
Hydrochloric Acid SCHEMBL1070020 0.99 ADAM10 (0.38) ADAM10ERBB2MMP1PIM1ABHD6
Hydrochloric Acid SCHEMBL878457 0.99 ADAM10 (0.38) ADAM10ERBB2MMP1PIM1ABHD6
SCHEMBL8008160 0.89 ADAM10 (0.39) ADAM10ERBB2MMP1ABHD6DPP8
SCHEMBL8060188 0.86 DPP8 (0.43) ADAM10ERBB2MMP1PIM1ABHD6
SCHEMBL8193679 0.86 DPP8 (0.43) ADAM10ERBB2MMP1PIM1ABHD6
SCHEMBL8117948 0.85 ADAM10 (0.41) ADAM10ERBB2MMP1PIM1ABHD6
Hydrochloric Acid SCHEMBL4584873 0.85 DPP8 (0.42) ADAM10ERBB2MMP1PIM1ABHD6
SCHEMBL8262157 0.84 PIM1 (0.33) ADAM10ERBB2MMP1PIM1ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076278-B1 Macrocyclic HCV NS3 protease inhibitors MERCK SHARP & DOHME (US) 2015-05-06 EP disclosed