SCHEMBL1667731

SCHEMBL1667731

C/C=C(/C)c1c(C(N)=NO)c2cccnc2n1-c1ccc(O)cc1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 4/20 0.33
PIM1 P11309 4/20 0.33
CHEK1 O14757 3/20 0.33
CDK2 P24941 3/20 0.33
CSNK2A1 P68400 3/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
FEN1 P39748 1/20 0.32
USP14 P54578 1/20 0.32
REN P00797 1/20 0.31
PPARG P37231 1/20 0.30
KDM1A O60341 1/20 0.30
APP P05067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1667736 1.00 NTRK1 (0.33) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL1667729 1.00 NTRK1 (0.33) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL1667676 0.88 NTRK1 (0.34) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL1667677 0.88 NTRK1 (0.34) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL1668112 0.86 HSP90AA1 (0.41) HSP90AA1HSP90AB1FEN1USP14REN
SCHEMBL1668113 0.86 HSP90AA1 (0.41) HSP90AA1HSP90AB1FEN1USP14REN
SCHEMBL1668111 0.86 HSP90AA1 (0.41) HSP90AA1HSP90AB1FEN1USP14REN
SCHEMBL1077738 0.81 SMN1; SMN2 (0.33) PPARGKDM1A
SCHEMBL1077734 0.81 SMN1; SMN2 (0.33) PPARGKDM1A
SCHEMBL1667733 0.80 FEN1 (0.32) FEN1USP14PPARGAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed