SCHEMBL1667924

SCHEMBL1667924

COC1CN(Cc2ccc(Nc3nccc(-c4ccc(OC5CCN(C(=O)CO)C5)c(C#N)c4)n3)cc2)C1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 20/20 0.61
JAK2 O60674 10/20 0.61
IKBKE Q14164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12274803 1.00 TBK1 (0.61) TBK1JAK2IKBKE
SCHEMBL1669857 0.93 TBK1 (0.62) TBK1JAK2IKBKE
SCHEMBL13279947 0.91 TBK1 (0.57) TBK1JAK2IKBKE
SCHEMBL13279999 0.91 TBK1 (0.57) TBK1JAK2IKBKE
SCHEMBL1667116 0.91 TBK1 (0.61) TBK1JAK2IKBKE
SCHEMBL12277014 0.88 TBK1 (0.62) TBK1JAK2
SCHEMBL1667390 0.86 TBK1 (0.63) TBK1JAK2IKBKE
SCHEMBL1667387 0.86 TBK1 (0.63) TBK1JAK2IKBKE
SCHEMBL1667171 0.86 TBK1 (0.67) TBK1JAK2
SCHEMBL13279840 0.85 TBK1 (0.61) TBK1JAK2IKBKE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488503-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON Myrexis, Inc. (US) 2012-08-22 EP disclosed
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed