SCHEMBL1668002

SCHEMBL1668002

CCN1CCC(CCCOc2cc(Nc3nccc(-c4cccc(C#N)c4OC4CCOCC4)n3)ccc2OC)CC1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 20/20 0.48
IKBKE Q14164 13/20 0.48
JAK2 O60674 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1669856 0.88 TBK1 (0.61) TBK1IKBKE
SCHEMBL12521834 0.81 JAK2 (0.48) TBK1IKBKEJAK2
SCHEMBL12274108 0.80 TBK1 (0.66) TBK1IKBKEJAK2
SCHEMBL12274545 0.79 TBK1 (0.61) TBK1IKBKE
SCHEMBL1667594 0.78 TBK1 (0.60) TBK1IKBKEJAK2
SCHEMBL1667567 0.77 IKBKE (0.71) TBK1IKBKE
SCHEMBL17327589 0.76 TBK1 (0.57) TBK1IKBKEJAK2
SCHEMBL1669942 0.76 TBK1 (0.72) TBK1IKBKEJAK2
SCHEMBL12274386 0.74 TBK1 (0.65) TBK1IKBKEJAK2
SCHEMBL12801141 0.73 TBK1 (0.51) TBK1IKBKEJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed