SCHEMBL16684145

SCHEMBL16684145

N#Cc1ccc(OP(=O)(O)CNS(=O)(=O)c2cc3cc(OCCNC(=O)c4cccc(O)c4O)c(OCCN)cc3s2)cc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.33
HDAC6 Q9UBN7 2/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TRPV4 Q9HBA0 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
HDAC2 Q92769 1/20 0.31
PLA2G7 Q13093 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13022858 0.97 AR (0.35) ARHDAC6ALDH1A1LMNAGAA
SCHEMBL12979768 0.95 AR (0.34) ARHDAC6ALDH1A1LMNAGAA
SCHEMBL14943076 0.94 AR (0.33) ARHDAC6ALDH1A1LMNAGAA
SCHEMBL14943075 0.94 AR (0.33) ARHDAC6ALDH1A1LMNAGAA
SCHEMBL16684148 0.92 TRPV4 (0.33) ALDH1A1LMNAGAASMN1; SMN2TRPV4
SCHEMBL3483982 0.92 TRPV4 (0.33) ALDH1A1LMNAGAASMN1; SMN2TRPV4
SCHEMBL14942995 0.90 CYP1A2 (0.32) ARHDAC6ALDH1A1LMNAGAA
SCHEMBL16684158 0.90 CYP1A2 (0.32) ARHDAC6ALDH1A1LMNAGAA
SCHEMBL13021466 0.90 TRPV4 (0.33) ALDH1A1LMNAGAASMN1; SMN2TRPV4
SCHEMBL13031987 0.89 SLC22A12 (0.34) ARTRPV4PLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049200-B1 NOVEL INHIBITORS OF BETA-LACTAMASE METHYLGENE INC (CA) 2015-04-29 EP disclosed