SCHEMBL16684161

SCHEMBL16684161

N#Cc1ccc(OP(=O)(O)CNS(=O)(=O)c2nc3cc(OCCCN)c(OCCCN)cc3s2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
TRPV4 Q9HBA0 9/20 0.35
SLC22A12 Q96S37 3/20 0.35
CACNA1B Q00975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14931225 0.96 CA1 (0.37) CA1CA2TRPV4SLC22A12
SCHEMBL14931332 0.89 SLC22A12 (0.33) CA1CA2TRPV4SLC22A12
SCHEMBL12979525 0.86 EGLN1 (0.32) CA1CA2TRPV4SLC22A12
SCHEMBL14943083 0.85 TRPV4 (0.36) TRPV4
SCHEMBL3480751 0.84 TRPV4 (0.35) TRPV4
SCHEMBL3480039 0.84 TRPV4 (0.35) TRPV4
SCHEMBL14931259 0.84 TRPV4 (0.34) TRPV4SLC22A12
SCHEMBL14943073 0.83 TRPV4 (0.35) TRPV4
SCHEMBL13032060 0.82 TRPV4 (0.36) TRPV4
SCHEMBL13031985 0.81 TRPV4 (0.36) TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049200-B1 NOVEL INHIBITORS OF BETA-LACTAMASE METHYLGENE INC (CA) 2015-04-29 EP disclosed