SCHEMBL16684690

SCHEMBL16684690

NC(=O)C1CCN(c2ccc3c(c2)CCCC3)C1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 10/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
PDK2 Q15119 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
KDM2B Q8NHM5 1/20 0.42
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16695100 1.00 NOTUM (0.47) NOTUMSMN1; SMN2PDK2NPC1RAB9A
SCHEMBL16695146 1.00 NOTUM (0.47) NOTUMSMN1; SMN2PDK2NPC1RAB9A
SCHEMBL16695240 0.87 NOTUM (0.62) NOTUM
SCHEMBL16695078 0.84 NOTUM (0.43) NOTUMPDK2
SCHEMBL16695065 0.84 NOTUM (0.43) NOTUMPDK2
SCHEMBL16695411 0.83 MAPT (0.47) NOTUMSMN1; SMN2PDK2NPC1RAB9A
SCHEMBL30263140 0.77 NOTUM (0.76) NOTUM
SCHEMBL16695120 0.76 NOTUM (0.54) NOTUM
SCHEMBL2636602 0.76 NOTUM (0.54) NOTUM
SCHEMBL16695072 0.76 DPP4 (0.52) NOTUMSMN1; SMN2PDK2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-A1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BioMarin Pharmaceutical Inc. (US) 2016-09-07 EP disclosed
WO-2015065937-A1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARMACEUTICAL INC. (US) 2015-05-07 WO disclosed