SCHEMBL16687553

SCHEMBL16687553

O=C(NCCc1cccc(CF)c1)c1sccc1Nc1ccnc2[nH]ccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 2/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
RAB9A P51151 5/20 0.38
NPC1 O15118 4/20 0.38
NAMPT P43490 1/20 0.37
TNNI3K Q59H18 1/20 0.36
CDK8 P49336 2/20 0.36
NEK1 Q96PY6 1/20 0.36
AKT1 P31749 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HTT P42858 1/20 0.35
ROCK1 Q13464 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
USP28 Q96RU2 2/20 0.34
USP25 Q9UHP3 2/20 0.34
MAPK8 P45983 1/20 0.34
MAPK10 P53779 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12901011 0.91 SNCA (0.41) BTKJAK2JAK1TYK2NPC1
SCHEMBL12901008 0.89 SMN1; SMN2 (0.48) BTKJAK2JAK1TYK2RAB9A
SCHEMBL19390620 0.89 RAB9A (0.43) BTKJAK2JAK1TYK2RAB9A
SCHEMBL12901005 0.89 CDK8 (0.47) JAK2JAK1TNNI3KCDK8AKT1
SCHEMBL12900654 0.88 ROCK1 (0.47) RAB9ANAMPTROCK1ADORA2AADORA2B
SCHEMBL12900697 0.86 HDAC2 (0.42) JAK2JAK1TYK2RAB9ANPC1
SCHEMBL12901013 0.85 NPC1 (0.43) JAK2JAK1TYK2RAB9ANPC1
SCHEMBL12901006 0.85 HDAC2 (0.40) JAK2JAK1TYK2RAB9ANPC1
SCHEMBL19390444 0.83 MAPT (0.46) JAK2JAK1TYK2RAB9ANPC1
SCHEMBL12900374 0.83 AKT1 (0.39) JAK2JAK1TYK2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9023847-B2 Azaheterocyclic compounds MERCK PATENT GMBH (DE) 2015-05-05 US disclosed