SCHEMBL16690686

SCHEMBL16690686

COC(=O)c1ccc(C(=O)c2c(CCCc3ccccc3)ccc(OC)c2F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.45
HPGD P15428 1/20 0.45
MGLL Q99685 1/20 0.44
CYP4F2 P78329 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PDE4D Q08499 3/20 0.42
ACHE P22303 1/20 0.42
POLB P06746 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
MEN1 O00255 1/20 0.42
PLAAT3 P53816 1/20 0.42
PLAAT5 Q96KN8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18044447 0.80 ATM (0.55) HPGDNPC1RAB9AKMT2ALMNA
SCHEMBL6261633 0.75 CYP4A11 (0.60) CYP4A11HPGDMGLLCYP4F2NPC1
SCHEMBL16334096 0.73 AKT1 (0.49) HPGDNPC1RAB9AKMT2ALMNA
SCHEMBL16690694 0.73 TDP1 (0.47) HPGDNPC1RAB9AKMT2ALMNA
SCHEMBL5061105 0.73 MAPT (0.45) CYP4A11NPC1RAB9AKMT2ALMNA
SCHEMBL2404460 0.73 CYP4A11 (0.73) CYP4A11MGLLCYP4F2NPC1RAB9A
SCHEMBL4630496 0.72 EGFR (0.45) NPC1RAB9AKMT2ALMNACA1
SCHEMBL8322717 0.71 PTGER1 (0.77) CYP4A11HPGDMGLLCYP4F2RAB9A
SCHEMBL1928912 0.71 TSHR (0.67) CYP4A11HPGDMGLLCYP4F2NPC1
SCHEMBL18010709 0.71 PDE4D (0.48) HPGDRAB9AKMT2ALMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015062555-A1 COMPOUND HAVING HIGHER INHIBITION OF PROTEIN KINASE G ACTIVITY AND PREPARATION METHOD THEREFOR 天津键凯科技有限公司 2015-05-07 WO disclosed