SCHEMBL1669355

SCHEMBL1669355

Nc1ncnc2c1nc(Sc1cc3c(cc1-c1ncco1)CCO3)n2CCC1CCN(CC=O)CC1

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.64
HSP90AB1 P08238 20/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1669353 0.88 HSP90AA1 (0.67) HSP90AA1HSP90AB1
SCHEMBL11908459 0.85 HSP90AA1 (0.70) HSP90AA1HSP90AB1
SCHEMBL1669199 0.83 HSP90AA1 (0.54) HSP90AA1HSP90AB1
SCHEMBL11909924 0.81 HSP90AA1 (0.56) HSP90AA1HSP90AB1
SCHEMBL1669530 0.81 HSP90AA1 (0.54) HSP90AA1HSP90AB1
SCHEMBL1670480 0.79 HSP90AB1 (0.51) HSP90AA1HSP90AB1
SCHEMBL3520073 0.79 HSP90AA1 (0.84) HSP90AA1HSP90AB1
SCHEMBL3520350 0.78 HSP90AA1 (1.00) HSP90AA1HSP90AB1
SCHEMBL1670755 0.78 HSP90AA1 (0.75) HSP90AA1HSP90AB1
SCHEMBL3518285 0.77 HSP90AA1 (0.78) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486039-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS Sloan Kettering Institute For Cancer Research (US) 2012-08-15 EP disclosed
WO-2011044394-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2011-04-14 WO disclosed