SCHEMBL16694479

SCHEMBL16694479

O=C1c2cc3c(cc2C2(CC2)N1CCC1CCN(Cc2ccccc2F)CC1)OCO3

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16694438 0.91
SCHEMBL16694123 0.90
SCHEMBL15599167 0.89
SCHEMBL15599182 0.89 CXCR4 (0.48)
SCHEMBL16886956 0.89
SCHEMBL16694166 0.89
SCHEMBL15598886 0.88 ACHE (0.52)
Hydrochloric Acid SCHEMBL16694401 0.87 ACHE (0.51)
SCHEMBL15599106 0.87 MCHR1 (0.45)
SCHEMBL15598768 0.87

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2871184-B1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF ZHEJIANG HISUN PHARM CO LTD (CN) 2017-09-06 EP claimed
US-9346818-B2 Benzodioxole derivative and preparation method and use thereof ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2016-05-24 US claimed
US-20150191480-A1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2015-07-09 US claimed
EP-2871184-A1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF Zhejiang Hisun Pharmaceutical Co. Ltd. (CN) 2015-05-13 EP claimed
EP-2871184-B1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF ZHEJIANG HISUN PHARM CO LTD (CN) 2017-09-06 EP disclosed
EP-2871184-B1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF ZHEJIANG HISUN PHARM CO LTD (CN) 2017-09-06 EP disclosed
US-9346818-B2 Benzodioxole derivative and preparation method and use thereof ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2016-05-24 US disclosed
US-9346818-B2 Benzodioxole derivative and preparation method and use thereof ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2016-05-24 US disclosed
US-9346818-B2 Benzodioxole derivative and preparation method and use thereof ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2016-05-24 US disclosed
US-20150191480-A1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2015-07-09 US disclosed
US-20150191480-A1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2015-07-09 US disclosed
US-20150191480-A1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2015-07-09 US disclosed
EP-2871184-A1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF Zhejiang Hisun Pharmaceutical Co. Ltd. (CN) 2015-05-13 EP disclosed
EP-2871184-A1 BENZODIOXOLE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF Zhejiang Hisun Pharmaceutical Co. Ltd. (CN) 2015-05-13 EP disclosed