SCHEMBL16696019

SCHEMBL16696019

CS(=O)(=O)CCCn1c(CCl)nc(=O)c2cc(Cl)ccc21

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.41
HRH4 Q9H3N8 1/20 0.39
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
NUDT1 P36639 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29606736 0.86 BACE1 (0.48) NUDT1BACE1
SCHEMBL15415657 0.86 BACE1 (0.48) NUDT1BACE1
Hydrochloric Acid SCHEMBL17074940 0.85 BACE1 (0.47) NUDT1BACE1
SCHEMBL16695998 0.81 PLK1 (0.45) CHEK1GABRA1GABRG2GABRB3GABRA5
SCHEMBL16696077 0.80 ALDH1A1 (0.45) CHEK1GABRA1GABRG2GABRB3GABRA5
SCHEMBL15415545 0.79 KMT2A (0.46) NUDT1BACE1
SCHEMBL16696060 0.78 PSEN1 (0.40) CHEK1PSEN1PSEN2APH1BNCSTN
SCHEMBL16696030 0.77 CYP3A4 (0.45)
SCHEMBL15908535 0.76 TBXA2R (0.37) ALDH1A1LMNA
SCHEMBL15650536 0.76 BACE1 (0.53) NUDT1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015065336-A1 RESPIRATORY SYNCYTIAL VIRUS INHIBITORS MEDIVIR AB (SE) 2015-05-07 WO disclosed