SCHEMBL1669714

SCHEMBL1669714

CS(=O)(=O)N1CCC(CCn2c(Sc3cc4c(cc3I)CCC4=O)nc3c(N)ncnc32)C1

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.60
HSP90AB1 P08238 20/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670196 0.87 HSP90AA1 (0.73) HSP90AA1HSP90AB1
SCHEMBL11908775 0.86 HSP90AA1 (0.62) HSP90AA1HSP90AB1
SCHEMBL11909679 0.86 HSP90AA1 (0.56) HSP90AA1HSP90AB1
SCHEMBL1670456 0.86 HSP90AB1 (0.57) HSP90AA1HSP90AB1
SCHEMBL1669266 0.83 HSP90AA1 (0.52) HSP90AA1HSP90AB1
SCHEMBL13193752 0.82 HSP90AB1 (0.51) HSP90AA1HSP90AB1
SCHEMBL15609718 0.81 HSP90AB1 (0.53) HSP90AA1HSP90AB1
SCHEMBL1669367 0.81 HSP90AB1 (0.56) HSP90AA1HSP90AB1
SCHEMBL29580670 0.80 HSP90AB1 (0.53) HSP90AA1HSP90AB1
SCHEMBL13194184 0.80 HSP90AB1 (0.53) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3091019-B1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2019-04-03 EP disclosed
EP-3091019-A2 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS Sloan Kettering Institute For Cancer Research (US) 2016-11-09 EP disclosed
EP-2486039-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS Sloan Kettering Institute For Cancer Research (US) 2012-08-15 EP disclosed
WO-2011044394-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2011-04-14 WO disclosed