SCHEMBL1669948

SCHEMBL1669948

CN1C=CCc2ccc(N)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.41
KDM4E B2RXH2 6/20 0.41
RAD52 P43351 1/20 0.41
ALDH1A1 P00352 8/20 0.35
LMNA P02545 5/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
CASP1 P29466 1/20 0.35
ADRA2C P18825 2/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
GAA P10253 3/20 0.33
KMT2A Q03164 3/20 0.33
PTK2B Q14289 2/20 0.33
MEN1 O00255 2/20 0.33
THRB P10828 2/20 0.33
NR4A1 P22736 1/20 0.33
GFER P55789 1/20 0.32
ESR2 Q92731 1/20 0.32
ATAD2 Q6PL18 2/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12637619 0.79 ALDH1A1 (0.37) MAPTALDH1A1
SCHEMBL3999191 0.71 MAPT (0.44) MAPTKDM4ERAD52ALDH1A1LMNA
SCHEMBL3360819 0.68 MAPT (0.44) MAPTKDM4ERAD52ALDH1A1LMNA
Hydrochloric Acid SCHEMBL31174158 0.67 MAPT (0.44) MAPTKDM4ERAD52ALDH1A1LMNA
Hydrochloric Acid SCHEMBL28709952 0.67 MAPT (0.44) MAPTKDM4ERAD52ALDH1A1LMNA
Hydrochloric Acid SCHEMBL27970719 0.67 MAPT (0.44) MAPTKDM4ERAD52ALDH1A1LMNA
Hydrochloric Acid SCHEMBL29386046 0.67 MAPT (0.44) MAPTKDM4ERAD52ALDH1A1LMNA
SCHEMBL520908 0.67 BRD4 (0.51) MAPTKDM4ERAD52ALDH1A1ADRA2C
SCHEMBL29240610 0.66 MAPT (0.45) MAPTKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL10511110 0.64 DRD1 (0.44) MAPTKDM4ELMNAHTTDRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486009-A1 2H-PYRROL-5-AMINE DERIVATIVES AS ALPHA ADRENERGIC RECEPTOR MODULATORS Allergan, Inc. (US) 2012-08-15 EP disclosed
WO-2011044229-A1 2H-PYRROL-5-AMINE DERIVATIVES AS ALPHA ADRENERGIC RECEPTOR MODULATORS ALLERGAN, INC. (US) 2011-04-14 WO disclosed