SCHEMBL16705118

SCHEMBL16705118

N#Cc1cccc(Sc2ccc3c(c2)COB3O)c1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 16/20 0.62
PDE4A P27815 11/20 0.62
PDE4C Q08493 11/20 0.62
PDE4D Q08499 11/20 0.62
PDE3A Q14432 2/20 0.53
CHRM1 P11229 1/20 0.53
ADRA1A P35348 1/20 0.53
PDE1A P54750 1/20 0.53
PDE3B Q13370 1/20 0.53
PDE7A Q13946 1/20 0.53
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16705119 0.90 PDE4B (0.53) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL16586497 0.88 PDE4B (0.64) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL5583384 0.80 PDE4B (0.71) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL596680 0.80 PDE4B (0.71) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL10172478 0.79 PDE4B (0.50) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL16705121 0.79 PDE4B (0.57) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL16705115 0.77 PDE4B (0.53) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL5583207 0.77 PDE4B (1.00) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL595173 0.77 PDE4B (1.00) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL26425601 0.77 PDE4B (0.62) PDE4BPDE4APDE4CPDE4DPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9029353-B2 Boron-containing small molecules as anti-inflammatory agents ANACOR PHARMACEUTICALS, INC. (US) 2015-05-12 US disclosed