SCHEMBL16705121

SCHEMBL16705121

N#Cc1ccccc1Sc1ccc2c(c1)COB2O

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 13/20 0.57
PDE4A P27815 8/20 0.57
PDE4C Q08493 7/20 0.57
PDE4D Q08499 7/20 0.57
PDE3A Q14432 2/20 0.46
CHRM1 P11229 1/20 0.46
ADRA1A P35348 1/20 0.46
PDE1A P54750 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE7A Q13946 1/20 0.46
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
AR P10275 3/20 0.39
PGR P06401 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16705120 0.90 PDE4B (0.48) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL10172481 0.85 AR (0.41) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL16586497 0.79 PDE4B (0.64) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL10172483 0.79 AR (0.41) PDE4BPDE4APDE4CPDE4DAR
SCHEMBL16705118 0.79 PDE4B (0.62) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL10217430 0.76 PDE4B (0.48) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL595613 0.72 PDE4B (1.00) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL5583343 0.72 PDE4B (1.00) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL12431297 0.71 PDE4B (0.76) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL24478326 0.70 CA1 (0.57) PDE4BPDE4APDE4CPDE4DPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9029353-B2 Boron-containing small molecules as anti-inflammatory agents ANACOR PHARMACEUTICALS, INC. (US) 2015-05-12 US disclosed