SCHEMBL16705120

SCHEMBL16705120

N#Cc1ccccc1Sc1ccc2c(c1)B(O)OC2

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.48
PDE4A P27815 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
CA1 P00915 6/20 0.44
CA2 P00918 6/20 0.44
CA12 O43570 5/20 0.43
CA9 Q16790 5/20 0.43
CA4 P22748 1/20 0.41
PGR P06401 1/20 0.39
AR P10275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16705121 0.90 PDE4B (0.57) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL10172483 0.86 AR (0.41) PDE4BPDE4APDE4CPDE4DPGR
SCHEMBL2280789 0.81 CA1 (0.47) CA1CA2CA12CA9CA4
SCHEMBL10172481 0.80 AR (0.41) PDE4BPDE4APDE4CPDE4DPGR
SCHEMBL16705115 0.79 PDE4B (0.53) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL16705119 0.79 PDE4B (0.53) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL596081 0.78 CA1 (0.54) CA1CA2CA12CA9CA4
SCHEMBL5528362 0.78 CA1 (0.54) CA1CA2CA12CA9CA4
SCHEMBL10217430 0.76 PDE4B (0.48) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL2287109 0.76 CA1 (0.44) CA1CA2CA12CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9029353-B2 Boron-containing small molecules as anti-inflammatory agents ANACOR PHARMACEUTICALS, INC. (US) 2015-05-12 US disclosed