SCHEMBL1670754

SCHEMBL1670754

CC(O)C(NC(C)(C)C)n1c(Sc2cc3c(cc2I)CCC3)nc2c(N)ncnc21

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 10/20 0.43
HSP90AB1 P08238 9/20 0.43
HSP90B1 P14625 7/20 0.43
HSP90AA1 P07900 7/20 0.43
TRAP1 Q12931 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670750 0.78 ERBB2 (0.49) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL18203411 0.75 HSP90AB1 (0.69) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL20860787 0.75 HSP90AB1 (0.52) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL15609147 0.75 HSP90AB1 (0.52) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL24377246 0.74 HSP90AB1 (0.61) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL17771103 0.74 HSP90AB1 (0.66) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL20548149 0.74 HSP90B1 (0.37) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL1669699 0.74 ERBB2 (0.69) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL1669814 0.74 HSP90AA1 (0.75) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1
SCHEMBL13193759 0.73 HSP90AB1 (0.54) ERBB2HSP90AB1HSP90B1HSP90AA1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011044394-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2011-04-14 WO disclosed