SCHEMBL20548149

SCHEMBL20548149

Cc1cnc(-c2cc3c(cc2Sc2nc4c(N)ncnc4n2C(NC(C)C)C(C)O)CCC3)o1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90B1 P14625 11/20 0.37
HSP90AA1 P07900 13/20 0.34
HSP90AB1 P08238 11/20 0.34
ERBB2 P04626 3/20 0.34
TRAP1 Q12931 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11909583 0.81 HSP90AA1 (0.42) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL11904625 0.79 HSP90AA1 (0.58) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL11904860 0.78 HSP90AA1 (0.46) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL1669554 0.76 HSP90AB1 (0.54) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL1669324 0.75 HSP90AB1 (0.53) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL1670754 0.74 ERBB2 (0.43) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL11908898 0.74 HSP90AA1 (0.48) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL11908349 0.73 HSP90AA1 (0.44) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL28461213 0.71 HSP90B1 (0.45) HSP90B1HSP90AA1HSP90AB1ERBB2TRAP1
SCHEMBL1670182 0.71 HSP90AA1 (0.51) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111683658-A Multi-protein complex inhibitor therapy for traumatic brain injury and sequelae thereof 萨缪斯治疗股份有限公司 2020-09-18 CN disclosed
EP-3641751-A2 EPICHAPEROME INHIBITOR THERAPY FOR TRAUMATIC BRAIN INJURY AND SEQUELAE THEREOF Samus Therapeutics, Inc. (US) 2020-04-29 EP disclosed
EP-3615008-A1 HSP90 INHIBITOR ORAL FORMULATIONS AND RELATED METHODS Samus Therapeutics, Inc. (US) 2020-03-04 EP disclosed
WO-2018237211-A2 EPICHAPEROME INHIBITOR THERAPY FOR TRAUMATIC BRAIN INJURY AND SEQUELAE THEREOF SAMUS THERAPEUTICS, INC. (US) 2018-12-27 WO disclosed
WO-2018200534-A1 HSP90 INHIBITOR ORAL FORMULATIONS AND RELATED METHODS SAMUS THERAPEUTICS, INC. (US) 2018-11-01 WO disclosed