SCHEMBL16719331

SCHEMBL16719331

O=S(=O)(Nc1ccc2cc[nH]c2c1)c1ccc2cc[nH]c2c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.78
CYP19A1 P11511 1/20 0.78
HTR6 P50406 1/20 0.78
HDAC3 O15379 2/20 0.60
HDAC4 P56524 2/20 0.60
HDAC1 Q13547 2/20 0.60
HDAC7 Q8WUI4 2/20 0.60
HDAC2 Q92769 2/20 0.60
HDAC10 Q969S8 2/20 0.60
HDAC11 Q96DB2 2/20 0.60
HDAC8 Q9BY41 2/20 0.60
HDAC6 Q9UBN7 2/20 0.60
HDAC9 Q9UKV0 2/20 0.60
HDAC5 Q9UQL6 2/20 0.60
KMT2A Q03164 3/20 0.51
ATIC P31939 1/20 0.50
MEN1 O00255 2/20 0.48
ALDH1A1 P00352 1/20 0.47
PKM P14618 1/20 0.46
PKLR P30613 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517779 0.88 ESR1 (0.62) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL5820194 0.88 ESR1 (0.74) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL4881882 0.86 ESR1 (0.76) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL16719349 0.85 ESR1 (0.59) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL3037102 0.85 ESR1 (0.80) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL16719422 0.84 ESR1 (0.59) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL16719591 0.84 ESR1 (0.62) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL16719616 0.84 ESR1 (0.70) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL7137662 0.83 MEN1 (0.66) ESR1CYP19A1HTR6HDAC3HDAC4
SCHEMBL19329860 0.82 HTR6 (0.62) ESR1CYP19A1HTR6HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed