SCHEMBL16720482

SCHEMBL16720482

Oc1cncc(-n2cccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.42
CHRNA4 P43681 2/20 0.42
POLB P06746 3/20 0.35
APLNR P35414 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ALK Q9UM73 1/20 0.33
VHL P40337 1/20 0.33
ELOC Q15369 1/20 0.33
ELOB Q15370 1/20 0.33
MAPT P10636 1/20 0.33
HSD17B1 P14061 1/20 0.32
ENPP2 Q13822 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
MIF P14174 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30201408 0.74 MAPT (0.52) POLBKDM4EALDH1A1ALKMAPT
SCHEMBL12369610 0.74 CHRNB2 (0.44) CHRNB2CHRNA4POLBKDM4EHSD17B10
SCHEMBL5659919 0.74 CHRNB2 (0.47) CHRNB2CHRNA4POLBKDM4EALDH1A1
SCHEMBL30811828 0.74 CHRNB2 (0.44) CHRNB2CHRNA4POLBKDM4EMAPT
SCHEMBL17819718 0.74 VHL (0.52) CHRNB2CHRNA4POLBKDM4EALK
SCHEMBL31456616 0.74 CA12 (0.40) CHRNB2CHRNA4MAPTHSD17B1
SCHEMBL1423044 0.72 HCAR2 (0.48) CHRNB2CHRNA4POLBKDM4EALDH1A1
SCHEMBL29465138 0.70 CYP2E1 (0.54) CHRNB2CHRNA4CYP3A4CYP2A6
SCHEMBL29464651 0.70 CHRNB2 (0.42) CHRNB2CHRNA4POLBAPLNRKDM4E
SCHEMBL3819587 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed