SCHEMBL16722331

SCHEMBL16722331

Cc1ccc(C(CCCOc2ccc(CN3CC(C(=O)O)C3)cc2)c2cccc(Cl)c2)cc1C

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 17/20 0.59
S1PR1 P21453 15/20 0.59
S1PR3 Q99500 4/20 0.54
LTK P29376 1/20 0.51
TAOK1 Q7L7X3 1/20 0.51
HTR2A P28223 1/20 0.48
KCNH2 Q12809 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
PDGFRA P16234 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16722011 0.90 S1PR1 (0.49) S1PR5S1PR1S1PR3
SCHEMBL16722437 0.90 S1PR5 (0.54) S1PR5S1PR1S1PR3PDGFRA
SCHEMBL15191985 0.89 S1PR5 (0.56) S1PR5S1PR1S1PR3LTKTAOK1
SCHEMBL16722188 0.88 S1PR5 (0.56) S1PR5S1PR1S1PR3LTKTAOK1
SCHEMBL16722014 0.88 S1PR5 (0.54) S1PR5S1PR1S1PR3
SCHEMBL16722681 0.88 S1PR5 (0.56) S1PR5S1PR1S1PR3PDGFRA
SCHEMBL16722661 0.86 S1PR5 (0.56) S1PR5S1PR1S1PR3HTR2AKCNH2
SCHEMBL15191748 0.86 S1PR5 (0.55) S1PR5S1PR1S1PR3LTKTAOK1
SCHEMBL15191692 0.86 S1PR5 (0.57) S1PR5S1PR1S1PR3LTKTAOK1
SCHEMBL16722391 0.85 S1PR5 (0.54) S1PR5S1PR1S1PR3HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015073547-A1 DISUBSTITUTED PHENOXY AZETIDINE DERIVATIVES AS SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR MODULATORS ALLERGAN, INC. (US) 2015-05-21 WO claimed
WO-2015073547-A1 DISUBSTITUTED PHENOXY AZETIDINE DERIVATIVES AS SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR MODULATORS ALLERGAN, INC. (US) 2015-05-21 WO disclosed
WO-2015073547-A1 DISUBSTITUTED PHENOXY AZETIDINE DERIVATIVES AS SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR MODULATORS ALLERGAN, INC. (US) 2015-05-21 WO disclosed