SCHEMBL16728429

SCHEMBL16728429

CO[C@]12CN(Cc3ccccc3)C[C@H]1CN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RORC P51449 11/20 0.43
OPRD1 P41143 1/20 0.43
OPRK1 P41145 1/20 0.43
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
GPR119 Q8TDV5 1/20 0.41
STS P08842 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2D6 P10635 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20274569 1.00 RORC (0.43) RORCOPRD1OPRK1JAK2JAK1
SCHEMBL14805534 1.00 RORC (0.43) RORCOPRD1OPRK1JAK2JAK1
SCHEMBL16728431 0.89 RORC (0.42) RORCOPRD1OPRK1JAK2JAK1
SCHEMBL14805536 0.89 RORC (0.42) RORCOPRD1OPRK1JAK2JAK1
SCHEMBL14801926 0.86 CYP2D6 (0.42) KDM4EALDH1A1CYP2D6
SCHEMBL14801928 0.86 CYP2D6 (0.42) KDM4EALDH1A1CYP2D6
SCHEMBL14801925 0.86 CYP2D6 (0.42) KDM4EALDH1A1CYP2D6
SCHEMBL24276430 0.84 RORC (0.46) RORCOPRD1OPRK1JAK2JAK1
SCHEMBL18668635 0.84 RORC (0.46) RORCOPRD1OPRK1JAK2JAK1
SCHEMBL29597428 0.84 RORC (0.46) RORCOPRD1OPRK1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9040547-B2 Pyrrolopyrimidine and purine derivatives PFIZER INC. (US) 2015-05-26 US disclosed