SCHEMBL16740929

SCHEMBL16740929

COc1cccc(C(=O)[C@H](C)CN(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.54
CES1 P23141 1/20 0.54
CHRNA1 P02708 1/20 0.52
CHRNG P07510 1/20 0.52
CHRNB1 P11230 1/20 0.52
CHRNB2 P17787 1/20 0.52
SLC6A2 P23975 1/20 0.52
CHRNB4 P30926 1/20 0.52
CHRNA3 P32297 1/20 0.52
CHRNA4 P43681 1/20 0.52
SLC6A3 Q01959 1/20 0.52
CHRND Q07001 1/20 0.52
PARP1 P09874 1/20 0.51
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
CTNNB1 P35222 1/20 0.47
WNT3A P56704 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL670521 1.00 CES2 (0.54) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL670522 1.00 CES2 (0.54) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL12393864 1.00 CES2 (0.54) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL30181112 1.00 CES2 (0.54) CES2CES1CHRNA1CHRNGCHRNB1
Hydrochloric Acid SCHEMBL671151 0.99 CES2 (0.53) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL670343 0.89 NPC1 (0.44) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL2411119 0.87 TP53 (0.49) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL670344 0.87 TP53 (0.49) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL30515227 0.87 TP53 (0.49) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL10855246 0.84 KDM4E (0.54) MEN1KMT2ACYP2D6HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4116288-A1 RACEMIZATION OF (S) AND/OR (R)-3-(DIMETHYLAMINO)-1-(3-METHOXYPHENYL)-2-METHYLPROPAN-1- ONE AND ITS MIXTURES KRKA, d.d., Novo mesto (SI) 2023-01-11 EP disclosed
WO-2015075678-A1 A NOVEL PROCESS FOR THE PREPARATION OF 1-PHENYL-3-AMINOPROPANE DERIVATIVES UNIMARK REMEDIES LTD. (IN) 2015-05-28 WO disclosed