SCHEMBL1675259

SCHEMBL1675259

c1nc(N2CCNCC2)c2cc(-c3ccc4c(c3)OCO4)ccc2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 17/20 1.00
CYP3A4 P08684 17/20 1.00
CYP2C19 P33261 9/20 1.00
CYP2D6 P10635 9/20 1.00
LMNA P02545 7/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
CLK4 Q9HAZ1 11/20 0.75
USP2 O75604 7/20 0.75
ALDH1A1 P00352 6/20 0.75
MAPK1 P28482 4/20 0.75
HIF1A Q16665 2/20 0.75
HSD17B10 Q99714 7/20 0.66
KDM4E B2RXH2 5/20 0.63
MAPT P10636 4/20 0.63
HPGD P15428 2/20 0.63
HTT P42858 2/20 0.58
TSHR P16473 4/20 0.58
ALOX15 P16050 1/20 0.56
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1675322 0.88 CLK4 (0.78) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL1675378 0.87 CYP3A4 (0.77) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL2913230 0.83 CYP1A2 (0.71) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL1675346 0.81 CLK4 (0.68) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
Chlorobenzene SCHEMBL27644941 0.74 CYP1A2 (0.69) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL3852063 0.74 HTT (0.68) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL6785138 0.74 HTT (0.70) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL2922462 0.74 HTT (0.70) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL1675117 0.74 CLK4 (0.65) CYP1A2CYP3A4CYP2C19CYP2D6LMNA
SCHEMBL2797008 0.74 HTT (1.00) CYP1A2CYP3A4CYP2C19CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO claimed
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO disclosed