SCHEMBL1675355

SCHEMBL1675355

COc1ccc(CNc2ncnc3ccc(-c4ccc5c(c4)OCO5)cc23)c(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 17/20 1.00
CYP3A4 P08684 17/20 1.00
CYP2C19 P33261 16/20 1.00
CLK4 Q9HAZ1 15/20 1.00
CYP2D6 P10635 15/20 1.00
CYP2C9 P11712 13/20 1.00
ALDH1A1 P00352 12/20 1.00
HSD17B10 Q99714 11/20 1.00
TSHR P16473 10/20 1.00
USP2 O75604 10/20 1.00
MAPK1 P28482 10/20 1.00
MEN1 O00255 5/20 1.00
KMT2A Q03164 5/20 1.00
ALOX15 P16050 4/20 1.00
LMNA P02545 12/20 0.79
HIF1A Q16665 5/20 0.79
PDE5A O76074 1/20 0.69
KDM4E B2RXH2 2/20 0.69
TDP1 Q9NUW8 1/20 0.69
CLK1 P49759 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1675333 0.88 CYP2D6 (1.00) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL1675031 0.83 CYP1A2 (1.00) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL30140903 0.82 PDE5A (1.00) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL678438 0.82 PDE5A (1.00) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL31066913 0.82 PDE5A (1.00) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL1584878 0.80 CYP1A2 (0.73) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL1675362 0.79 CLK1 (0.82) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL1675139 0.78 CLK4 (0.74) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL1675357 0.78 CLK4 (1.00) CYP1A2CYP3A4CYP2C19CLK4CYP2D6
SCHEMBL4866306 0.78 CYP1A2 (0.73) CYP1A2CYP3A4CYP2C19CLK4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO claimed
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO disclosed