SCHEMBL16760397

SCHEMBL16760397

COc1cc2c(Cl)ncnc2cc1OCc1cccnc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.67
EPHA2 P29317 3/20 0.67
EPHB4 P54760 2/20 0.67
FLT1 P17948 2/20 0.67
ENPP1 P22413 3/20 0.61
RET P07949 1/20 0.56
KIF5B P33176 1/20 0.56
PDPK1 O15530 1/20 0.51
ERBB2 P04626 1/20 0.49
PDGFRB P09619 3/20 0.48
PDGFRA P16234 3/20 0.48
PDE10A Q9Y233 1/20 0.48
HTT P42858 2/20 0.47
LMNA P02545 2/20 0.47
RAF1 P04049 1/20 0.47
MAPK1 P28482 1/20 0.47
ATM Q13315 1/20 0.47
KDM4E B2RXH2 1/20 0.46
EGFR P00533 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29631520 0.86 ENPP1 (0.68) KDRENPP1RETHTTLMNA
SCHEMBL297514 0.86 ENPP1 (0.68) KDRENPP1RETHTTLMNA
SCHEMBL295891 0.86 ENPP1 (0.68) KDRENPP1RETHTTLMNA
Hydrochloric Acid SCHEMBL156332 0.85 ENPP1 (0.67) ENPP1PDGFRBPDGFRAHTTLMNA
Hydrochloric Acid SCHEMBL28041015 0.85 ENPP1 (0.67) ENPP1PDGFRBPDGFRAHTTLMNA
Hydrochloric Acid SCHEMBL28102763 0.85 ENPP1 (0.67) ENPP1PDGFRBPDGFRAHTTLMNA
SCHEMBL7205078 0.85 ENPP1 (0.67) KDREPHA2EPHB4FLT1ENPP1
SCHEMBL906880 0.81 EPHA2 (1.00) KDREPHA2EPHB4FLT1ERBB2
SCHEMBL8857758 0.79 ENPP1 (0.56) ENPP1HTTLMNAMAPK1ATM
SCHEMBL364049 0.79 ENPP1 (0.81) KDRFLT1ENPP1RETLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015079251-A1 QUINAZOLINE COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2015-06-04 WO disclosed
WO-2015079251-A1 QUINAZOLINE COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2015-06-04 WO disclosed