SCHEMBL16768664

SCHEMBL16768664

C=C(NCCc1nc2ccccc2s1)C(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2C19 P33261 2/20 0.51
HSD17B10 Q99714 2/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
HIF1A Q16665 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.47
ALOX15 P16050 2/20 0.47
HTT P42858 2/20 0.47
RAB9A P51151 1/20 0.46
POLB P06746 3/20 0.45
ATM Q13315 1/20 0.45
UBE2T Q9NPD8 1/20 0.45
ASIC3 Q9UHC3 1/20 0.45
ALDH1A1 P00352 4/20 0.45
PDE10A Q9Y233 2/20 0.44
SLC13A5 Q86YT5 1/20 0.44
GAA P10253 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16133681 0.84 SMN1; SMN2 (0.53) HPGDCYP1A2CYP2C19HSD17B10CYP3A4
SCHEMBL17050824 0.79 SMN1; SMN2 (0.57) HPGDCYP1A2CYP2C19SMN1; SMN2ALOX15
SCHEMBL16136346 0.77 HPGD (0.55) HPGDCYP1A2CYP2C19HSD17B10SMN1; SMN2
SCHEMBL7435843 0.76 UBE2T (0.56) HPGDCYP1A2CYP2C19HSD17B10CYP3A4
SCHEMBL18381211 0.75 SLC13A5 (0.56) HPGDCYP1A2CYP2C19HSD17B10CYP3A4
SCHEMBL11683409 0.75 CA12 (0.50) HPGDCYP1A2CYP2C19HSD17B10CYP3A4
SCHEMBL17481133 0.74 HPGD (0.69) HPGDCYP1A2CYP2C19HSD17B10CYP3A4
SCHEMBL23374667 0.74 UBE2T (0.53) HPGDCYP1A2CYP2C19HSD17B10CYP3A4
SCHEMBL19372016 0.74 UBE2T (0.70) HPGDCYP1A2CYP2C19HSD17B10CYP3A4
SCHEMBL24198727 0.73 HPGD (0.63) HPGDCYP1A2CYP2C19HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9776996-B2 Substituted 6,5-fused bicyclic heteroaryl compounds Epizyme, Inc. (US) 2017-10-03 US disclosed
US-9045477-B2 Substituted 6,5-fused bicyclic heteroaryl compounds Epizyme, Inc. (US) 2015-06-02 US disclosed