SCHEMBL16768698

SCHEMBL16768698

C=C(NCc1cn(C)cn1)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
MTOR P42345 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
HPGDS O60760 1/20 0.39
OGA O60502 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
SLC6A2 P23975 1/20 0.34
HTR1D P28221 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
MAPK1 P28482 1/20 0.34
EGLN2 Q96KS0 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
METTL3 Q86U44 1/20 0.32
SYK P43405 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12935908 0.81 HPGDS (0.44) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL12257137 0.75 CYP2C9 (0.50) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL28712747 0.75 HPGD (0.44) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL12332384 0.75 NPSR1 (0.49) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL2937818 0.75 HPGDS (0.46) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL25836690 0.74 KDM4E (0.46) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL1487971 0.73
SCHEMBL30894898 0.73 CYP2C9 (0.55) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL16768682 0.72
SCHEMBL12964153 0.72 HPGDS (0.44) CYP2C9TSHRCYP2C19MTORHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9045477-B2 Substituted 6,5-fused bicyclic heteroaryl compounds Epizyme, Inc. (US) 2015-06-02 US disclosed