SCHEMBL16774672

SCHEMBL16774672

[CH2]Cc1cnc2cc[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.44
APP P05067 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.40
BRAF P15056 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PRKCI P41743 1/20 0.32
MAPK1 P28482 2/20 0.31
FAAH O00519 1/20 0.31
QPCT Q16769 1/20 0.31
MAPT P10636 1/20 0.31
RAD52 P43351 1/20 0.31
ACKR3 P25106 1/20 0.30
SYK P43405 1/20 0.30
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30
NAMPT P43490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4400758 0.81 BRD4 (0.44) BRD4APPPIK3C3BRAFKDM4E
SCHEMBL14637827 0.79 CDK8 (0.40) BRD4APPPIK3C3BRAFKDM4E
SCHEMBL14637826 0.79 BRD4 (0.39) BRD4APPPIK3C3BRAFKDM4E
SCHEMBL19682171 0.77 BRD4 (0.41) BRD4APPPIK3C3BRAFKDM4E
SCHEMBL24600122 0.74 BRD4 (0.44) BRD4APPPIK3C3KDM4EALDH1A1
SCHEMBL28007340 0.73 FGFR1 (0.39) BRD4APPPIK3C3MAPK1SYK
SCHEMBL15058223 0.72 AHR (0.47) BRD4APPPIK3C3KDM4EALDH1A1
SCHEMBL28036822 0.72 QPCTL (0.40) BRD4
SCHEMBL1269027 0.71 TYR (0.45) BRD4APPPIK3C3KDM4EALDH1A1
SCHEMBL15058364 0.71 AHR (0.45) BRD4APPPIK3C3BRAFKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2734516-B1 ARYLPYRAZOLE ETHERS AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE BOEHRINGER INGELHEIM INT (DE) 2015-06-17 EP claimed