SCHEMBL28036822

SCHEMBL28036822

Fc1cccc(Cc2cnc3cc[nH]c3c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCTL Q9NXS2 1/20 0.40
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
SNCA P37840 2/20 0.38
DAO P14920 1/20 0.38
BRD4 O60885 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
DBH P09172 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
ERBB3 P21860 1/20 0.36
ERBB4 Q15303 1/20 0.36
TAAR1 Q96RJ0 2/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KIT P10721 1/20 0.36
P2RX7 Q99572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28195435 0.79 QPCTL (0.55) QPCTL
SCHEMBL28215219 0.76 PIK3C3 (0.48) QPCTLBRD4TAAR1
SCHEMBL28037237 0.76 AHR (0.58) HTR2CHTR2BDAODBHTAAR1
SCHEMBL28047821 0.73 AHR (0.42) HTR2CHTR2BDAOHCAR2DBH
SCHEMBL15058364 0.72 AHR (0.45) BRD4
SCHEMBL3300303 0.72 TAAR1 (0.60) DAOHCAR2TAAR1SMN1; SMN2
SCHEMBL16774672 0.72 BRD4 (0.44) BRD4
SCHEMBL4400758 0.72 BRD4 (0.44) BRD4L3MBTL1
SCHEMBL28047883 0.71 SNCA (0.41) HTR2CHTR2BSNCADAOHCAR2
SCHEMBL28195437 0.71 QPCTL (0.46) QPCTLHTR2CHTR2BSNCADAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189481-A Pyridine cdk9 kinase inhibitors ABBVIE INC 2015-12-23 CN disclosed
CN-105026393-A Cdk9 kinase inhibitors ABBVIE INC 2015-11-04 CN disclosed