SCHEMBL16784064

SCHEMBL16784064

CCCCn1c(NS(=O)(=O)c2ccccc2)c(S(=O)(=O)c2ccc(C)cc2)c2nccnc21

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.75
MAPT P10636 11/20 0.75
KDM4E B2RXH2 10/20 0.75
HPGD P15428 9/20 0.75
GAA P10253 7/20 0.75
BLM P54132 6/20 0.75
KMT2A Q03164 6/20 0.75
SAE1 Q9UBE0 6/20 0.75
UBA2 Q9UBT2 6/20 0.75
HTT P42858 6/20 0.75
MEN1 O00255 5/20 0.75
SMN1; SMN2 Q16637 5/20 0.75
RXFP1 Q9HBX9 4/20 0.75
L3MBTL1 Q9Y468 4/20 0.75
THRB P10828 4/20 0.75
NPSR1 Q6W5P4 4/20 0.75
PLEC Q15149 3/20 0.75
UBE2I P63279 3/20 0.75
NSD2 O96028 3/20 0.75
TDP2 O95551 2/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16772922 0.85 KDM4E (0.55) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL15256901 0.85 KDM4E (1.00) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL15256904 0.79 KDM4E (0.89) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL15256919 0.79 KDM4E (0.68) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL19742978 0.78 SAE1 (0.70) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL15256869 0.71 KDM4E (0.75) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL15256897 0.70 HPGD (1.00) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL15032608 0.70 ALDH1A1 (0.71) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL6981812 0.70 SAE1 (0.89) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL6981187 0.66 KDM4E (1.00) ALDH1A1MAPTKDM4EHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9045483-B2 Inhibition of small ubiquitin-like modifier enzymes with substituted pyrrolo[2,3-b]quinoxalines CITY OF HOPE (US) 2015-06-02 US disclosed