SCHEMBL1679258

SCHEMBL1679258

CS(=O)(=O)NCc1cccc(Br)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.54
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 2/20 0.47
TAAR1 Q96RJ0 2/20 0.47
BRD4 O60885 1/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
MAPT P10636 1/20 0.46
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.45
RECQL P46063 1/20 0.45
NFATC1 O95644 1/20 0.45
NR3C1 P04150 1/20 0.45
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
CARM1 Q86X55 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23732903 0.84 CYP19A1 (0.53) CYP19A1CYP1A2CYP2D6CYP2C19TAAR1
SCHEMBL14431548 0.83 TAAR1 (0.62) CYP1A2CYP2D6CYP2C19TAAR1POLB
SCHEMBL23732923 0.83 CYP19A1 (0.51) CYP19A1CYP1A2CYP2D6CYP2C19TAAR1
SCHEMBL2529923 0.81 CYP19A1 (0.50) CYP19A1CYP1A2CYP2D6CYP2C19TAAR1
SCHEMBL13462548 0.80 CYP19A1 (0.51) CYP19A1BRD4KMT2AKDM4EPOLB
SCHEMBL8265344 0.80 CYP19A1 (0.56) CYP19A1CYP1A2CYP2D6CYP2C19BRD4
SCHEMBL27811793 0.80 CYP19A1 (0.51) CYP19A1BRD4KMT2AKDM4EPOLB
SCHEMBL23703127 0.79 CYP19A1 (0.51) CYP19A1KMT2AMEN1PKMRAB9A
SCHEMBL3102964 0.79 CYP19A1 (0.49) CYP19A1BRD4KMT2AKDM4EPOLB
SCHEMBL1542377 0.79 CYP19A1 (0.61) CYP19A1BRD4KMT2AKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12195490-B2 STRAD-binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-01-14 US disclosed
CN-115916966-A STRAD binding agents and uses thereof 加利福尼亚大学董事会 2023-04-04 CN disclosed
WO-2021155004-A1 STRAD-BINDING AGENTS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-08-05 WO disclosed
US-7923573-B2 Benzene compound having 2 or more substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-04-12 US disclosed
US-20080004301-A1 Benzene Compound Having 2 or More Substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-01-03 US disclosed
EP-1806332-A1 BENZENE COMPOUND HAVING 2 OR MORE SUBSTITUENTS Daiichi Sankyo Company, Limited (JP) 2007-07-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12195490-B2 STRAD-binding agents and uses thereof STRAP, STRA6, PLAUR CYP19A1 4547/4885CYP1A2 4758/4885CYP2D6 4584/4885
US-20080004301-A1 Benzene Compound Having 2 or More Substituents NR1H2, NR1H3, NCOR2 CYP19A1 118/4885CYP1A2 187/4885CYP2D6 552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.