SCHEMBL1542377

SCHEMBL1542377

CS(=O)(=O)NCc1cccc(N)c1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.61
BRD4 O60885 1/20 0.47
PRMT1 Q99873 1/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.45
RECQL P46063 1/20 0.45
KMT2A Q03164 1/20 0.45
TP53 P04637 1/20 0.44
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
NAMPT P43490 1/20 0.44
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 1/20 0.43
CA12 O43570 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
NFATC1 O95644 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14206309 0.85 CYP19A1 (0.50) CYP19A1PRMT1POLBKMT2ATP53
SCHEMBL15651955 0.84 CYP19A1 (0.59) CYP19A1PRMT1KDM4EKMT2ATP53
SCHEMBL11666038 0.83 PRMT1 (0.57) CYP19A1PRMT1POLBMAOAMAOB
SCHEMBL1684383 0.82 CA1 (0.51) CYP19A1BRD4KDM4EPOLBTSHR
SCHEMBL2495774 0.81 CYP19A1 (0.56) CYP19A1PRMT1KMT2AMAOAMAOB
SCHEMBL8265344 0.80 CYP19A1 (0.56) CYP19A1BRD4KDM4EPOLBTSHR
SCHEMBL13462548 0.80 CYP19A1 (0.51) CYP19A1BRD4KDM4EPOLBTSHR
SCHEMBL27811793 0.80 CYP19A1 (0.51) CYP19A1BRD4KDM4EPOLBTSHR
SCHEMBL1679258 0.79 CYP19A1 (0.54) CYP19A1BRD4KDM4EPOLBTSHR
SCHEMBL3102964 0.79 CYP19A1 (0.49) CYP19A1BRD4KDM4EPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC 2010-04-01 US claimed
WO-2010034671-A1 PYRINE OR PYRAZINE DERIVATIVES FOR TREATING HCV F. HOFFMANN-LA ROCHE AG (CH) 2010-04-01 WO claimed
EP-4334298-B1 UREA DERIVATIVES WHICH CAN BE USED TO TREAT CANCER SCORPION THERAPEUTICS INC (US) 2026-02-18 EP disclosed
US-20250250259-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. 2025-08-07 US disclosed
US-12312341-B2 Methods for treating cancer SCORPION THERAPEUTICS, INC. (US) 2025-05-27 US disclosed
EP-3617213-B1 THIENO[3,2-D]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY FOR PROTEIN KINASES HANMI PHARMACEUTICAL CO LTD (KR) 2025-02-19 EP disclosed
US-20240400543-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. 2024-12-05 US disclosed
US-20240300939-A1 UREA DERIVATIVES WHICH CAN BE USED TO TREAT CANCER SCORPION THERAPEUTICS, INC. 2024-09-12 US disclosed
US-12084434-B2 Methods for treating cancer SCORPION THERAPEUTICS, INC. (US) 2024-09-10 US disclosed
US-20240158376-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. 2024-05-16 US disclosed
CN-117813293-A Urea derivatives useful for the treatment of cancer 蝎子疗法股份有限公司 2024-04-02 CN disclosed
WO-2011077171-A1 4-PHENYLAMINO-PYRIMIDINE DERIVATIVES HAVING PROTEIN KINASE INHIBITOR ACTIVITY VICHEM CHEMIE KUTATÓ KFT. (HU) 2011-06-30 WO disclosed
WO-2011077171-A1 4-PHENYLAMINO-PYRIMIDINE DERIVATIVES HAVING PROTEIN KINASE INHIBITOR ACTIVITY VICHEM CHEMIE KUTATÓ KFT. (HU) 2011-06-30 WO disclosed
EP-2307372-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-04-13 EP disclosed
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC 2010-04-01 US disclosed
WO-2010034671-A1 PYRINE OR PYRAZINE DERIVATIVES FOR TREATING HCV F. HOFFMANN-LA ROCHE AG (CH) 2010-04-01 WO disclosed
WO-2010010017-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-01-28 WO disclosed
US-20100021423-A1 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC 2010-01-28 US disclosed
US-20070054916-A1 Aryl nitrogen-containing bicyclic compounds and methods of use AMGEN INC. 2007-03-08 US disclosed
US-20070054916-A1 Aryl nitrogen-containing bicyclic compounds and methods of use AMGEN INC. 2007-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240300939-A1 UREA DERIVATIVES WHICH CAN BE USED TO TREAT CANCER PIK3CA, PIK3CG, PIK3CD CYP19A1 498/4885BRD4 4438/4885PRMT1 418/4885
US-20240158376-A1 METHODS FOR TREATING CANCER PIK3CA, PTEN, BRCA1 CYP19A1 255/4885BRD4 2997/4885PRMT1 1705/4885
US-12312341-B2 Methods for treating cancer PIK3CA, PTEN, BRCA1 CYP19A1 255/4885BRD4 2997/4885PRMT1 1705/4885
US-20070054916-A1 Aryl nitrogen-containing bicyclic compounds and methods of use MAP3K1, MAP3K5, MAP3K2 CYP19A1 171/4885BRD4 395/4885PRMT1 421/4885
US-20250250259-A1 METHODS FOR TREATING CANCER PIK3CA, PTEN, BRCA1 CYP19A1 255/4885BRD4 2997/4885PRMT1 1705/4885
US-20240400543-A1 METHODS FOR TREATING CANCER PIK3CA, PTEN, BRCA1 CYP19A1 255/4885BRD4 2997/4885PRMT1 1705/4885
US-12084434-B2 Methods for treating cancer PIK3CA, PTEN, BRCA1 CYP19A1 255/4885BRD4 2997/4885PRMT1 1705/4885
US-20100021423-A1 Heterocyclic antiviral compounds POLR2A, RRM2B, RRP1B CYP19A1 1594/4885BRD4 998/4885PRMT1 241/4885
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS EIF2AK2, POLR2A, HCCS CYP19A1 1679/4885BRD4 1086/4885PRMT1 1231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.