SCHEMBL16794896

SCHEMBL16794896

Cc1c(-c2cccc(-c3nnnn3C)c2)c2[nH]c3ccccc3c2[nH]c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.38
PADI4 Q9UM07 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
NQO2 P16083 1/20 0.36
ACLY P53396 1/20 0.35
PARP1 P09874 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA1 P30542 1/20 0.34
MAPK14 Q16539 1/20 0.34
CDK4 P11802 2/20 0.34
CCND1 P24385 2/20 0.34
CHEK1 O14757 1/20 0.34
WEE1 P30291 1/20 0.34
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
NR1I3 Q14994 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16814244 0.80 NQO2 (0.36) NPSR1PADI4KDM4EALDH1A1NQO2
SCHEMBL16814364 0.78 SERPINE1 (0.49) ADORA3ADORA1CDK4CCND1CCNE2
SCHEMBL16795016 0.78 PARP1 (0.39) NPSR1PADI4SMN1; SMN2KDM4EALDH1A1
SCHEMBL16814348 0.76 MDM2 (0.39) NPSR1PADI4KDM4EALDH1A1NQO2
SCHEMBL16814487 0.76 NQO2 (0.38) PADI4NQO2PARP1MAPK14CHEK1
SCHEMBL16814570 0.76 CYP11B1 (0.57) NPSR1PADI4SMN1; SMN2KDM4EALDH1A1
SCHEMBL16794875 0.76 NTRK1 (0.37) NPSR1PADI4SMN1; SMN2KDM4EALDH1A1
SCHEMBL16814275 0.75 NQO2 (0.38) NPSR1PADI4KDM4EALDH1A1NQO2
SCHEMBL16795035 0.75 NQO2 (0.42) NPSR1PADI4KDM4EALDH1A1NQO2
SCHEMBL16794852 0.75 NQO2 (0.38) NPSR1PADI4KDM4EALDH1A1NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088564-A1 P2X4 RECEPTOR MODULATING COMPOUNDS SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed
WO-2015088564-A1 P2X4 RECEPTOR MODULATING COMPOUNDS SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed