Bromide

Bromide

SCHEMBL1680033

Br.CCOc1ccc2c(C(=O)c3ccc(OCCN4CCCCC4)cc3)c(-c3ccc(OC)cc3)sc2c1

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A known ✓ P08913 1/20 0.71
ADRB3 known ✓ P13945 1/20 0.71
ADRA2B known ✓ P18089 1/20 0.71
ADRA2C known ✓ P18825 1/20 0.71
ACHE known ✓ P22303 1/20 0.71
SLC6A2 known ✓ P23975 1/20 0.71
ADRA1D known ✓ P25100 1/20 0.71
SLC6A4 known ✓ P31645 1/20 0.71
ADRA1A known ✓ P35348 1/20 0.71
SLC6A3 known ✓ Q01959 1/20 0.71
SIGMAR1 known ✓ Q99720 1/20 0.71
ESR1 P03372 18/20 0.88
ESR2 Q92731 18/20 0.88
ENPP3 O14638 2/20 0.76
ENPP1 P22413 1/20 0.76
MEN1 O00255 2/20 0.71
ALDH1A1 P00352 2/20 0.71
LMNA P02545 2/20 0.71
TP53 P04637 2/20 0.71
CYP3A4 P08684 2/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1680060 0.99 ESR1 (0.90) ESR1ESR2ENPP3ENPP1MEN1
SCHEMBL11209650 0.95 ESR1 (0.82) ESR1ESR2ENPP3MEN1ALDH1A1
Bromide SCHEMBL1665326 0.95 ESR1 (0.98) ESR1ESR2ENPP3ENPP1MEN1
SCHEMBL11188522 0.94 ESR1 (0.90) ESR1ESR2ENPP3ENPP1MEN1
SCHEMBL1665661 0.94 ESR1 (1.00) ESR1ESR2ENPP3ENPP1MEN1
Hydrochloric Acid SCHEMBL2495864 0.93 ESR1 (1.00) ESR1ESR2ENPP3ENPP1MEN1
SCHEMBL7632970 0.93 ESR1 (0.98) ESR1ESR2ENPP3ENPP1MEN1
Hydrochloric Acid SCHEMBL1665332 0.93 ESR1 (1.00) ESR1ESR2ENPP3ENPP1MEN1
SCHEMBL6663935 0.93 ESR1 (0.98) ESR1ESR2ENPP3ENPP1MEN1
SCHEMBL6595860 0.92 ESR1 (0.96) ESR1ESR2ENPP3ENPP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011047878-A2 A PROCESS FOR PREPARING BENZO[B]THIOPHENE DERIVATIVES HEXAL AKTIENGESELLSCHAFT (DE) 2011-04-28 WO disclosed