SCHEMBL16800730

SCHEMBL16800730

C#Cc1cccc(Nc2ncnn3cc(C(=O)O)c(C)c23)c1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.60
CSNK2A2 P19784 1/20 0.51
CSNK2B P67870 1/20 0.51
CSNK2A1 P68400 1/20 0.51
MAP2K1 Q02750 1/20 0.49
MAPK14 Q16539 5/20 0.48
EGFR P00533 3/20 0.48
ERBB2 P04626 2/20 0.48
AURKA O14965 1/20 0.48
RPS6KB1 P23443 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16800568 0.88 MAP2K1 (0.64) KDRMAP2K1MAPK14EGFRERBB2
SCHEMBL16800731 0.83 EGFR (0.52) KDREGFRERBB2AURKARPS6KB1
SCHEMBL5739243 0.82 KDR (0.60) KDRMAP2K1MAPK14EGFRERBB2
SCHEMBL4042333 0.80 KDR (0.75) KDRMAP2K1MAPK14EGFRERBB2
SCHEMBL28749813 0.80 KDR (0.58) KDRMAP2K1MAPK14EGFRERBB2
SCHEMBL16800829 0.80 KDR (0.49) KDRMAPK14EGFRERBB2AURKA
SCHEMBL12728722 0.79 KDR (0.62) KDRCSNK2A2CSNK2BCSNK2A1MAP2K1
SCHEMBL5516114 0.79 KDR (0.80) KDREGFR
SCHEMBL7530745 0.78 KDR (0.70) KDRMAP2K1MAPK14EGFRERBB2
SCHEMBL4053778 0.78 KDR (0.78) KDRMAP2K1MAPK14EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015081783-A1 PYRROLO[2,1-F][1,2,4]TRIAZINE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 江苏奥赛康药业股份有限公司 2015-06-11 WO disclosed