SCHEMBL5739243

SCHEMBL5739243

Cc1c(C(=O)O)cn2ncnc(Nc3cccc(NS(C)(=O)=O)c3)c12

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 0.60
MAP2K1 Q02750 1/20 0.49
EGFR P00533 3/20 0.48
ERBB2 P04626 2/20 0.48
MAPK14 Q16539 6/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051959 0.90 KDR (0.75) KDRMAP2K1EGFRERBB2MAPK14
SCHEMBL7583147 0.86 MAPK14 (0.58) KDREGFRMAPK14
SCHEMBL5740244 0.82 KDR (0.54) KDRMAP2K1EGFRERBB2MAPK14
SCHEMBL28749813 0.82 KDR (0.58) KDRMAP2K1EGFRERBB2MAPK14
SCHEMBL16800730 0.82 KDR (0.60) KDRMAP2K1EGFRERBB2MAPK14
SCHEMBL12728722 0.79 KDR (0.62) KDRMAP2K1EGFRMAPK14
SCHEMBL5516114 0.79 KDR (0.80) KDREGFR
SCHEMBL7530745 0.78 KDR (0.70) KDRMAP2K1EGFRERBB2MAPK14
SCHEMBL4053778 0.78 KDR (0.78) KDRMAP2K1EGFRERBB2MAPK14
SCHEMBL4044821 0.77 MAPK14 (0.69) KDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed