SCHEMBL1683000

SCHEMBL1683000

NCCOc1cccc(Cl)c1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.57
TP53 P04637 2/20 0.54
ALDH1A1 P00352 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
TSHR P16473 1/20 0.54
CYP2C19 P33261 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
HTR1B P28222 1/20 0.52
TAAR1 Q96RJ0 3/20 0.47
PNMT P11086 1/20 0.47
MAPK1 P28482 1/20 0.46
RAB9A P51151 1/20 0.46
GAA P10253 2/20 0.46
HTT P42858 1/20 0.46
DHFR P00374 2/20 0.45
DPP4 P27487 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1290535 0.98 KDM4E (0.61) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL14830658 0.90 ALDH1A1 (0.57) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL7968991 0.87 TDP1 (0.54) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL1032880 0.83 KDM4E (0.68) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
Hydrochloric Acid SCHEMBL6492504 0.82 KDM4E (0.72) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL13744588 0.81 KDM4E (0.53) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL10359841 0.80 TSHR (0.68) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL15473216 0.80 ALDH1A1 (0.54) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL28043167 0.80 ALDH1A1 (0.54) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL2206657 0.80 ALDH1A1 (0.54) KDM4ETP53ALDH1A1SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012045729-A1 IMIDAZO [1, 2 -A] PYRIDINE AND PYRAZOLO [1, 5 -A] PYRIDINE DERIVATIVES AS TRPV1 ANTAGONISTS GLAXO GROUP LIMITED (GB) 2012-04-12 WO disclosed