SCHEMBL16836089

SCHEMBL16836089

CC(C)(O)c1ncccc1C1=CCN(C(=O)O)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
GRM5 P41594 3/20 0.42
GRM1 Q13255 3/20 0.42
PDK4 Q16654 1/20 0.42
CHEK1 O14757 3/20 0.41
MAP4K4 O95819 3/20 0.41
PIM1 P11309 3/20 0.41
PRKACA P17612 3/20 0.41
CLK2 P49760 3/20 0.41
GSK3B P49841 3/20 0.41
CDK5 Q00535 3/20 0.41
PRKAA1 Q13131 3/20 0.41
ROCK1 Q13464 3/20 0.41
DYRK1A Q13627 3/20 0.41
CLK4 Q9HAZ1 3/20 0.41
CHEK2 O96017 2/20 0.41
PRKCG P05129 2/20 0.41
CDK1 P06493 2/20 0.41
FGFR1 P11362 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30136907 0.86 PDK4 (0.59) GRM5GRM1PDK4CDK9PDE10A
SCHEMBL16836014 0.86 PDK4 (0.59) GRM5GRM1PDK4CDK9PDE10A
Hydrochloric Acid SCHEMBL31025163 0.85 PDK4 (0.58) GRM5GRM1PDK4CDK9PDE10A
SCHEMBL15286283 0.82 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2GRM5GRM1CHEK1
SCHEMBL17363102 0.80 SMN1; SMN2 (0.49) ALDH1A1SMN1; SMN2CHEK1MAP4K4PIM1
SCHEMBL2640481 0.80 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2GRM5GRM1CHEK1
SCHEMBL25571346 0.79 PDK4 (0.45) GRM5GRM1PDK4CDK9PDE10A
SCHEMBL17397683 0.79 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2PDK4CHEK1MAP4K4
SCHEMBL16992066 0.79 PDE10A (0.46) ALDH1A1SMN1; SMN2PDK4CHEK1MAP4K4
SCHEMBL22328949 0.76 GRM5 (0.59) GRM5GRM1PDK4PDE10AJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3083633-A1 SPIRO-OXAZOLONES F.HOFFMANN-LA ROCHE AG (CH) 2016-10-26 EP disclosed
WO-2015091411-A1 SPIRO-OXAZOLONES F. HOFFMANN-LA ROCHE AG (CH) 2015-06-25 WO disclosed